Andrographolide

Andrographolide bụ ngwaahịa botanical nke ewepụtara site na ahịhịa nke na-emekarị na China.Osisi ahụ nwere ọtụtụ akụkọ ihe mere eme eji eme ihe na TCM maka ọgwụgwọ ọrịa nke akụkụ okuku ume elu na ọrịa ndị ọzọ na-egbu egbu na ọrịa.Andrographis paniculata ewebata ma kụọ ya na Guangdong na ndịda Fujian na 50s.A na-eji ya agwọ ọrịa dị iche iche na-efe efe na ata agwọ.N'ime afọ ndị na-adịbeghị anya, a mụọla ihe ọkụkụ, ihe mejupụtara kemịkalụ, ọgwụ na akụkụ ahụike nke Andrographis paniculata na China.Andrographis paniculata bụ ọgwụ ọdịnala ndị China na-ejikarị eme ihe, nke nwere mmetụta nke ikpochapụ okpomọkụ na nsị, na-eme ka ọbara dị jụụ na detumescence.N'ụlọ ọgwụ, a na-ejikarị ya agwọ ọrịa nke akụkụ okuku ume iku ume, nnukwu ọnyụnyụ bacillary, gastroenteritis, oyi, ahụ ọkụ na ọbara mgbali elu.Site na mmụba nke mmetọ ọgwụ nje na mmeghachi omume ọjọọ, olu nke na-emepụta ọgwụ ọdịnala ndị China nwere ezigbo mmetụta nje na-eto eto.Andrographis paniculata, dị ka ọgwụ ọdịnala ndị China nwere mmetụta nje, ka ụlọ ọrụ na-emepụta ọgwụ anabatala ya nke ukwuu.

Amara ihe ọkụkụ Andrographis paniculata nwere ọtụtụ ọrụ ọgwụ.Andrographolide, isi ihe na-emepụta ihe na-emetụta ọrụ ọgwụ ya.Anyị mụrụ usoro cellular na ebumnuche nke ọgwụgwọ andrographolide mebere na ọrịa kansa mmadụ na sel mgbochi.Ọgwụ Andrographolide gbochiri mmụba in vitro nke ahịrị mkpụrụ ndụ etuto dị iche iche, na-anọchi anya ụdị ọrịa cancer dị iche iche.Ngwa ahụ na-arụ ọrụ anticancer kpọmkwem na mkpụrụ ndụ kansa site na njide okirikiri cell na G0 / G1 oge site na ntinye nke protein inhibitory p27 cell-cycle na mbelata okwu nke cyclin-based kinase 4 (CDK4).A na-egosipụta ọrụ immunostimulatory nke andrographolide site na mmụba nke lymphocytes na mmepụta nke interleukin-2.Andrographolide kwalitekwara mmepụta necrosis factor-alpha tumor na okwu akara CD, na-ebute mmụba cytotoxic nke lymphocytes megide mkpụrụ ndụ kansa, nke nwere ike inye aka maka ọrụ mgbochi ọrịa kansa na-apụtaghị ìhè.A na-akwadokwa ọrụ anticancer in vivo nke ogige ahụ megidere B16F0 melanoma syngenic na ụdị HT-29 xenograft.Nsonaazụ ndị a na-egosi na andrographolide bụ pharmacophore na-adọrọ mmasị nke nwere ọrụ anticancer na immunomodulatory na ya mere enwere ike imepụta ya dị ka onye na-ahụ maka ọgwụgwọ ọrịa kansa.


Oge nzipu: Jun-22-2021